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European Journal of Applied Sciences – Vol. 11, No. 3

Publication Date: June 25, 2023

DOI:10.14738/aivp.113.14483.

Hovhannisyan, S., Mashinyan, K. A., Torgomyan, A. L., & Hakobyan, G. (2023). Graphene Oxide: The Promising Potential in

Dentistry: A Review. European Journal of Applied Sciences, Vol - 11(3). 269-278.

Services for Science and Education – United Kingdom

Graphene Oxide: The Promising Potential in Dentistry: A Review

Hovhannisyan, S.

Department of prosthodontics,

Yerevan State Medical University after M. Heratsi, Armenia

Mashinyan, K. A.

Department of prosthodontics, Yerevan State Medical

University after M. Heratsi, Armenia

Torgomyan, A. L.

Department of Physiology,

Yerevan State Medical University after M. Heratsi, Armenia

Hakobyan, G.

Dept. of Oral and Maxillofacial Surgery

Yerevan State Medical University after M. Heratsi, Armenia

ABSTRACT

Objectives: In recent years the applications of graphene oxide (GO) have been

extensively studied in various fields of medicine, due to its antibacterial properties

and the ability to regenerate tissues. In dentistry, graphene oxide (GO) is also used

to complement existing materials due to its unique properties, however, research

on the use of graphene in dentistry is limited. What dictates a comprehensive

review of the literature on the prospects for the use of graphene in clinical dentistry.

In this review, we aim to highlight the potential of Graphene oxide, current

understanding, and knowledge gaps regarding the antimicrobial behavior and

biocompatibility of this materials. The purpose of this review article is to provide

an overview of the use of graphene oxide (GO) in dentistry. Methods: Bibliographic

databases PubMed, Embase, and Scopus were surveyed. The review focuses on the

areas of application of Graphene oxide (GO) in dentistry, mainly based on a review

of the most cited scientific papers in international peer-reviewed journals. Results:

Graphene oxide (GO) has a unique structure and properties that differentiate it

from other materials. Scope of application Graphene oxide (GO) broad in dentistry,

it is used in prosthetics and restorative dentistry to optimize polymers and

adhesives, dental implantology, to modify the surface of dental implants, to

optimize the osteogenic properties of engineered tissue scaffolds through both

surface and composite modifications, in periododntology and in endodontics

thanks to his antimicrobial behavior. Conclusion: From this review, it can be

concluded about the prospects for future developments, the use of Graphene in

dentistry. Graphene oxide (GO) has the potential for future clinical applications in

a variety of dental applications.

Keywords: Nanomaterials, biocompatibility dental materials, Graphene oxide.

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European Journal of Applied Sciences (EJAS) Vol. 11, Issue 3, June-2023

INTRODUCTION

Dental materials placed in the oral cavity must be non-cytotoxic and biocompatible, resistant

to mechanical stress. There is a strong trend towards the continuous development of dental

materials with improved properties. In the 21st century, nanotechnology plays an important

role in almost all areas of science, technology, medicine, including dentistry. Nanotechnology is

the art of creating a variety of materials with different properties and functions, which opens

up great prospects in the field of denetal materials science. Nanotechnology is usually referred

to as technology leading to the production of materials of nanometer size (10-9 microns).

Nanostructures contain nanoparticles of different sizes (zero, one-, two- and three- dimensional. 3 New materials based on nanomaterials have improved physicochemical and

mechanical properties in combination, which makes them excellent materials for some dental

procedures The use of nanotechnology in dentistry is wide and includes nanorobotics,

nanodiagnostics, nanomaterials, and thanks to these achievements, many dental problems are

solved for the better - from the diagnosis of dental diseases to more effective treatment

methods. It is clear that current developments in nanotechnology hold promising prospects for

all aspects of dentistry. This review presents a perspective advantage Graphene oxide (GO) in

dentistry. All the data and articles putted in this review are gathered from Google Scholar,

PubMed, and some dental databases. The use of Graphene oxide in dentistry is enormous and

includes prosthetics, endodontics, conservative and aesthetic dentistry, periodontics,

implantology, and regenerative dentistry. Physical and technological properties Graphene

Oxide (GO) Graphene oxide (GO) family nanomaterials was first obtained by Geim and

Novoselov in 2004 [1,2]. Graphene oxide (GO) include ultrathin graphite, multilayer graphene

(FLG), graphene oxide (GO; monolayer to multiple layers), reduced graphene oxide (rGO), and

graphene nanosheets (GNS). GO is one of the crystalline forms of carbon, which is a single

monolayer of sp2 hybridized orbitals in a tightly packed to a two-dimensional (2D) honeycomb

lattice, each carbon atom has three σ-bonds and an out-of-plane π-bond that can bind with

neighboring atoms [1]. The structure of GO consists of a single atom layer and functional groups

such as carboxylic acid, epoxide, and hydroxyl groups which could make it amphiphilic [3]. GO

can be produced by various approaches including chemical vapor deposition [4], mechanical

cleavage of graphite, and electrochemical exfoliation of graphite [5]. GO can be further wrapped

up to form zero-dimension (0D) nanomaterial like fullerenes, or rolled into nanotube (one

dimension, 1D), or manipulated into 3D graphite [6]. GO sheets exist in bi-layers and multi- layers (<10), each possessing unique properties. Further increasing the number of layers

significantly changes the properties of the material as a graphene stack with 10 layers behave

more like graphite [6], demonstrating that the interlayer structure and coupling between the

layers determinekey physical properties [7].

For instance, the stacking order, relative twist, and interlayer spacing govern the electronic,

optical, and mechanical properties of multi-layered graphene [8]. Additionally, graphene is a

free-standing two-dimensionally active carbon allotrope, where each carbon atom in the 2D

crystal is bonded to the three other adjacent carbon atoms forming a hexagonal aromatic

structure [8]. This specific structure and its periodicity result in unique electrical and

mechanical characteristics. The electron confinement in the orbitals are localized to

neighboring carbon atoms to create the covalent σ-bonds [9]. Graphene's unique physical

properties include hardness higher than diamond, elastic modulus as highas 1 TPa [10], thermal

conductivity almost 13 times higher than copper [11], and good optical transparency with

~97.7% transmittance [12].

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Hovhannisyan, S., Mashinyan, K. A., Torgomyan, A. L., & Hakobyan, G. (2023). Graphene Oxide: The Promising Potential in Dentistry: A Review.

European Journal of Applied Sciences, Vol - 11(3). 269-278.

URL: http://dx.doi.org/10.14738/aivp.113.14483.

GO has many unique physicochemical and biological properties [13]. Graphene can be easily

functionalized with bioactive compounds such as proteins, enzymes, drugs, growth factors, and

DNAvia physical interaction [14].

GO is highly biocompatible, can promote cell adhesion and proliferation, and can induce

directed stem cell differentiation [15,16].

Since there are several types of microorganisms in the oral cavity that cause caries and

periodontitis procedures in the oral cavityusing dental materials are susceptible to the action of

microbes, thereforeit is advisable to provide dental materials with antimicrobial properties.

ANTIBACTERIAL PROPERTIES GRAPHENE OXIDE (GO)

In the oral cavity, bacteria involved in caries formation are Streptococcus mutans, and bacteria

associated with periodontitis and root canal infections are Porphyromonas gingivalis and

Fusobacterium nucleatum.

GO in combination with other compounds, for example, the graphene / zinc oxide

nanocomposite, exhibits enhanced synergistic antimicrobial, antibiotic-film, and antiadhesive

activity against oral pathogens.

GO has been shown to have excellent antibacterial properties through a variety of mechanisms

[17,18].

Researchers have identified the basic mechanisms of the antimicrobial activity of Graphene

which includes physical and chemical effects.

Physical mechanism GO 's antimicrobial effect is caused by the fact that graphene materials

penetratethe cell membrane of microbes, causing leakage of intracellular substance, leading to

cell death. Thechemical antimicrobial effect of Graphene is caused by primary oxidative stress

mediated by ROS production. Excessive accumulation of intracellular ROS causes inactivation

of intracellular protein,lipid peroxidation and mitochondrial dysfunction, which in turn leads to

the gradual destruction of thecell membrane and, ultimately, cell death [19].

Lee et al. have created PMMA, including nano-sized graphene oxide (nGO), which has shown

antiadhesive effects against microbial species (C. albicans, E. coli, S. aureus and S. mutans) in

artificial saliva. They observed a persistent antimicrobial adhesive effect for up to 28 days [20].

Majority of studies find GO as most effective by damaging the microbial cells with mechanical

interaction of sharp edges as well as by the generating reactive oxygen species (ROS) [21].

The first study showed strong antimicrobial behavior of both GO and rGO by deactivating the

98.5%and 90% of Escherichia coli (E. coli) DH5α cells [22].

A study by He et al. evaluated the antibacterial activity of GO nanosheets against three common

types of bacteria Streptococci mutans - Porphyromonas gingivalis and Fusobacterium

nucleatum against oral pathogens and found that GO nanosheets are very effective in inhibiting

the growth of these pathogens. At a GO concentration of 40 μg / ml, the growth of P. gingivalis

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European Journal of Applied Sciences (EJAS) Vol. 11, Issue 3, June-2023

and F. nucleatum bacteriawas inhibited, while at a concentration of 80 μg / ml, GO completely

killed all S. mutans [23].

Subsequently, the broad-spectrum antimicrobial activity of GO was demonstrated by

evaluating the antimicrobial activity against the phytopathogen and fungal species [24].

Antibacterial role of nano-graphene oxide was investigated by Wu et al. Thus they investigated

whether the graphene oxide (GO) nanosheets could be used to enhance antibacterial activity of

ASwalR RNA for E. faecalis in periapical periodontitis. They showed that GO-PEI could

efficiently deliver the ASwalR plasmid into E. faecalis cell. GO-PEI-ASwalR significantly reduced

virulent- associated gene expressions. Furthermore, GO-PEI-ASwalR suppressed biofilm

aggregation and improved bactericidal effects [25].

GO also has the potential for drug delivery [26].

Properties such as biocompatibility and low toxicity of GO open up the scope of its application

for the delivery of therapeutic drugs in the environment of these drugs BMP-2 aspirin [27],

vancomycin

[28] and miRNA [29,30]. Many of the graphene-based drug/gene delivery systems such as

nanocomposites of GO with vascular endothelial growth factor (VEGF) or GO carrier containing

mitoxantrone have been developed as cardiac tissue regeneration systems or a therapeutic

treatment for tumors [31].

The antibacterial properties of GO can be useful for dentists in various industries.

The antibacterial properties of GO can be very helpful in suture fabrication. It has been

suggested thatcompared to conventional polyvinyl alcohol (PVA) fiber, which does not have

antimicrobial properties. A PVA matrix dispersed with mechanically exfoliated graphene

(MEG) exhibits a high antibacterial effect and thus effectively accelerates wound healing,

making PVA/MEG nanocompositefiber a promising new candidate for surgical sutures [32].

Further in-depth experimental studies are needed to further analyze the bactericidal effect of

graphenefor future clinical applications, especially with respect to dental pathogens, as these

in vivo studies are still in their infancy. Applications of Graphene Oxide (GO) in Bone Tissue

Engineering. Bone regeneration is a complex and dynamic physiological process that at the

macroscopic level includes local mechanical stability, environmental matrix and blood supply,

and microscopically includes the interaction of many cells, signaling molecules and effectors in

a spatio-temporal sequence. The bone graft materials substitute should have the following

characteristics:

1) good biocompatibility

2) suitable mechanical properties to ensure adequate durability;

3) porous structure or rough surface to facilitate the germination of cells and tissues;

4) favorable osteoconductivity and osteoinduction to stimulate the formation of new bone;

5) controlled degradability to match the rate of germination of new bone;

6) non-immunogenicity to ensure safe clinical use.

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Hovhannisyan, S., Mashinyan, K. A., Torgomyan, A. L., & Hakobyan, G. (2023). Graphene Oxide: The Promising Potential in Dentistry: A Review.

European Journal of Applied Sciences, Vol - 11(3). 269-278.

URL: http://dx.doi.org/10.14738/aivp.113.14483.

The extraordinary mechanical and electronic properties of graphene-based materials have

motivatedresearchers to use them in tissue engineering and regenerative medicine [33].

Graphene and its derivatives provide a new selection for enhancing the mechanical and surface

properties of biomaterials to regulate the cardiomyogenic, neurogenic, osteogenic and

cartilaginous abilities of stem cells [34].

It is obvious that with these key multifunctional properties, graphene derivatives have shown

their potential and became favorite materials for many biomedical scientists, to design new

materials or hybrid materials or coatings of these nanomaterials to existing biomedical devices

to overcome with the possibility of device associated infections.

Thanks to its unique characteristics, graphene quickly became a potential candidate for

biomedical use. Overall, grapheme-based materials hold great promise for application in

different fields of medicine, more specifically in dentistry [35].

Its mechanical properties, including strength, stiffness, and flexibility, make it one of the most

anticipated materials for bone engineering and may hold the promise of using Graphene in bone

regeneration.

Good electrical conductivity of GO can not only directly stimulate the osteogenic activity of cells,

butalso indirectly adsorb active factors, promoting bone formation [36].

Thus, the properties of GO fully meet the requirements of dentistry and tissue engineering.

Lee et al investigated the ability of graphene oxide (rGO) and hydroxyapatite (HAp) (rGO / HAp

NCs) to enhance osteogenesis of MC3T3-E1 preosteoblasts and new bone formation [37].

The following study conducted by Nizami et al assessed the efficacy of functionalized graphene

oxide(f-GO) nanocomposites on the decalcification of dentin, because dental caries of the root

surface is becoming one of the new problems in aged society [38]. GO-Ag and GO-Ag-CaF2

almost completelyinhibited S. mutans growth. However, they did not exhibit cytotoxicity to

epithelial cells except at the highest concentration (0.1 w/v%) of GO-Ag and GOAg-CaF2.

Furthermore, these f-GOnanocomposites exhibited less or no discoloration of dentin, although

commonly used silver diaminefluoride causes discoloration of dentin to black. Thus, these f-GO

nanocomposites are useful to protectdental caries on the tooth root that becomes a social

problem in aged society [39].

The study of osteogenic mechanisms can indicate the right direction for further research; then,

elucidating the mechanisms of degradation and metabolism will help to understand the space- time distribution of GD in vivo [40].

Ahn et al investigate the efects of mesoporous bioactive glass nanoparticle (MBN)/graphene

oxide (GO) composites on the mineralization ability and differentiation potential of human

dental pulp stemcells (hDPSCs) [41].